SCHEMBL9833613

SCHEMBL9833613

CC1(c2cccnc2)CSC(N)=N1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.49
KCNH2 Q12809 2/20 0.38
CTSD P07339 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5330236 0.82 BACE1 (0.70) BACE1KCNH2
SCHEMBL5052720 0.72 BACE1 (0.65) BACE1KCNH2
SCHEMBL10154760 0.71 BACE1 (0.49) BACE1KCNH2
SCHEMBL19839752 0.70 BACE1 (0.36) BACE1
SCHEMBL159063 0.69 HCAR2 (0.38) BACE1
SCHEMBL4134312 0.69 BACE1 (0.71) BACE1BACE2
SCHEMBL17033073 0.66 ALDH1A1 (0.41)
SCHEMBL16052004 0.66 BACE1 (0.51) BACE1KCNH2CTSDBACE2
SCHEMBL10154712 0.66 BACE1 (1.00) BACE1KCNH2
SCHEMBL13306647 0.66 BACE1 (1.00) BACE1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0234011-B1 4-(1,2,5,6-TETRAHYDRO-1-ALKYL-3-PYRIDINYL)-2-THIAZOLAMINES AND 4-(HEXAHYDRO-1-ALKYL-3-PYRIDINYL)-2-THIAZOLAMINES WARNER-LAMBERT COMPANY (US) 1991-09-18 EP disclosed