SCHEMBL159063

SCHEMBL159063

CC1(c2cccnc2)CC[N]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2A6 P11509 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.35
P2RX7 Q99572 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
VNN1 O95497 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17033073 0.78 ALDH1A1 (0.41) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL1865507 0.76 ALDH1A1 (0.42) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL12586110 0.74 P2RX7 (0.42) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL16590522 0.74 ALDH1A1 (0.40) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL246083 0.72 CHRNB2 (0.43) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL10283135 0.72 CHRM2 (0.40) OPRM1OPRL1CHRM2CHRM4CHRM5
SCHEMBL122354 0.71 HCAR2 (0.42) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL13139599 0.70 OPRM1 (0.41) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL24867577 0.69 ALDH1A1 (0.43) HCAR2OPRM1OPRL1CHRM2CHRM4
SCHEMBL11971740 0.69 ALDH1A1 (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611788-A2 NICOTINE COMPOUNDS AND ANALOGS THEREOF, SYNTHETIC METHODS OF MAKING COMPOUNDS, AND METHODS OF USE University of Florida Research Foundation, Incorporated (US) 2013-07-10 EP disclosed
WO-2012031220-A2 NICOTINE COMPOUNDS AND ANALOGS THEREOF, SYNTHETIC METHODS OF MAKING COMPOUNDS, AND METHODS OF USE UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2012-03-08 WO disclosed