SCHEMBL9833865

SCHEMBL9833865

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2cccc(Cl)c2)c2c1CSc1ccc(Cl)cc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CCNA1 P78396 1/20 0.38
RIPK1 Q13546 1/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
MAPT P10636 4/20 0.35
PIK3CD O00329 1/20 0.35
PIK3R2 O00459 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
PIK3R5 Q8WYR1 1/20 0.35
PIK3R3 Q92569 1/20 0.35
F10 P00742 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9316496 0.97 MEN1 (0.40) POLBMEN1KMT2ARIPK1MAPT
SCHEMBL9831040 0.96 RIPK1 (0.41) POLBMEN1KMT2ACCNA2CDK2
SCHEMBL9832082 0.94 MAPT (0.39) POLBCCNA2CDK2CCNA1RIPK1
SCHEMBL9832532 0.93 ALDH1A1 (0.42) POLBMEN1KMT2ARIPK1MAPT
SCHEMBL9833948 0.92 ALDH1A1 (0.40) POLBMEN1KMT2ARIPK1MAPT
SCHEMBL9833256 0.92 RIPK1 (0.39) POLBMEN1KMT2ACCNA2CDK2
SCHEMBL9832608 0.92 NPC1 (0.40) POLBMEN1KMT2ARIPK1MAPT
SCHEMBL9831199 0.91 MAPT (0.39) MEN1KMT2ACCNA2CDK2CCNA1
SCHEMBL9833062 0.91 TP53 (0.41) CCNA2CDK2CCNA1RIPK1MAPT
SCHEMBL9316263 0.90 RIPK1 (0.41) MEN1KMT2ACCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed