SCHEMBL9833256

SCHEMBL9833256

N#CC(C(=O)Nc1cccc(F)c1)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccc(Cl)cc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.39
KCNJ6 P48051 7/20 0.37
KCNJ3 P48549 7/20 0.37
KCNJ5 P48544 5/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
IKBKB O14920 3/20 0.36
HSP90AA1 P07900 1/20 0.35
GRIK1 P39086 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
PIK3CD O00329 1/20 0.34
PIK3R2 O00459 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
PIK3R5 Q8WYR1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831040 0.94 RIPK1 (0.41) RIPK1KCNJ6KCNJ3KCNJ5MEN1
SCHEMBL9832532 0.94 ALDH1A1 (0.42) RIPK1KCNJ6KCNJ3KCNJ5MEN1
SCHEMBL9833948 0.93 ALDH1A1 (0.40) RIPK1MEN1POLBKMT2AALDH1A1
SCHEMBL9316496 0.93 MEN1 (0.40) RIPK1KCNJ6KCNJ3KCNJ5MEN1
SCHEMBL9832144 0.92 RIPK1 (0.41) RIPK1KCNJ6KCNJ3KCNJ5ALDH1A1
SCHEMBL9833865 0.92 POLB (0.39) RIPK1KCNJ6KCNJ3KCNJ5MEN1
SCHEMBL9832608 0.91 NPC1 (0.40) RIPK1KCNJ6KCNJ3KCNJ5MEN1
SCHEMBL9316263 0.88 RIPK1 (0.41) RIPK1KCNJ6KCNJ3KCNJ5MEN1
SCHEMBL10571543 0.88 RIPK1 (0.42) RIPK1KCNJ6KCNJ3KCNJ5MEN1
SCHEMBL9523052 0.88 RIPK1 (0.37) RIPK1KCNJ6KCNJ3KCNJ5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP claimed
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed