SCHEMBL9834534

SCHEMBL9834534

CC(C)(C)OC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.80
CTSS P25774 1/20 0.80
CTSK P43235 1/20 0.80
MAPT P10636 4/20 0.70
GAA P10253 1/20 0.70
HTT P42858 1/20 0.70
CCKBR P32239 3/20 0.69
TP53 P04637 1/20 0.67
ACE P12821 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.65
LMNA P02545 1/20 0.65
TACR1 P25103 2/20 0.65
NMBR P28336 4/20 0.62
KCNT1 Q5JUK3 1/20 0.62
KLK5 Q9Y337 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8395025 0.92 CTSL (0.72) CTSLCTSSCTSKMAPTGAA
SCHEMBL8271104 0.92 CTSL (0.72) CTSLCTSSCTSKMAPTGAA
SCHEMBL9833490 0.91 CTSL (0.76) CTSLCTSSCTSKMAPTCCKBR
SCHEMBL27839975 0.91 CTSL (0.69) CTSLCTSSCTSKMAPTGAA
SCHEMBL30375072 0.90 CTSL (0.80) CTSLCTSSCTSKMAPTCCKBR
SCHEMBL17807348 0.90 CTSL (0.80) CTSLCTSSCTSKMAPTCCKBR
SCHEMBL8482904 0.89 MAPT (0.75) CTSLCTSSCTSKMAPTGAA
SCHEMBL8482130 0.89 CTSL (0.73) CTSLCTSSCTSKMAPTGAA
SCHEMBL15220151 0.89 CTSL (0.65) CTSLCTSSCTSKMAPTGAA
SCHEMBL6021511 0.89 CTSS (1.00) CTSLCTSSCTSKMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0442878-A4 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS 1991-10-23 EP disclosed
EP-0442878-A1 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1991-08-28 EP disclosed
WO-1989010355-A1 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1989-11-02 WO disclosed
EP-0336356-A2 Derivatives of tryptophan as CCK antagonists ABBOTT LABORATORIES (US) 1989-10-11 EP disclosed