SCHEMBL9833490

SCHEMBL9833490

CC(C)(C)OC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCc1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.76
CTSS P25774 1/20 0.76
CTSK P43235 1/20 0.76
NMBR P28336 8/20 0.75
BRS3 P32247 2/20 0.67
TACR3 P29371 1/20 0.67
TACR1 P25103 1/20 0.65
MAPT P10636 2/20 0.64
TP53 P04637 1/20 0.64
ACE P12821 1/20 0.64
CCKBR P32239 2/20 0.63
BCHE P06276 1/20 0.62
ACHE P22303 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
KMT2A Q03164 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9834534 0.91 CTSL (0.80) CTSLCTSSCTSKNMBRTACR1
SCHEMBL7521907 0.90 CTSL (0.67) CTSLCTSSCTSKNMBRTACR3
SCHEMBL15145364 0.89 CTSL (0.77) CTSLCTSSCTSKNMBRTACR3
SCHEMBL15145404 0.89 CTSL (0.77) CTSLCTSSCTSKNMBRTACR3
SCHEMBL12371623 0.88 NMBR (0.64) CTSLCTSSCTSKNMBRBRS3
SCHEMBL18879584 0.87 CTSL (0.74) CTSLCTSSCTSKNMBRTACR3
SCHEMBL17884340 0.87 CTSL (0.74) CTSLCTSSCTSKNMBRTACR3
SCHEMBL30375072 0.87 CTSL (0.80) CTSLCTSSCTSKTACR3TACR1
SCHEMBL17807348 0.87 CTSL (0.80) CTSLCTSSCTSKNMBRTACR3
SCHEMBL8613263 0.87 CCKBR (0.68) CTSLCTSSCTSKNMBRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0442878-A4 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS 1991-10-23 EP disclosed
EP-0442878-A1 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1991-08-28 EP disclosed
WO-1989010355-A1 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1989-11-02 WO disclosed
EP-0336356-A2 Derivatives of tryptophan as CCK antagonists ABBOTT LABORATORIES (US) 1989-10-11 EP disclosed