SCHEMBL9834814

SCHEMBL9834814

CC1(C)OC(=O)C(c2cccc(C(F)(F)F)c2)=C1N

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
BRD4 O60885 1/20 0.44
XDH P47989 1/20 0.43
BACE1 P56817 2/20 0.42
CTSD P07339 1/20 0.42
NOTUM Q6P988 1/20 0.42
IKBKB O14920 1/20 0.41
PGR P06401 1/20 0.41
HCAR3 P49019 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
KIF11 P52732 1/20 0.39
RXRA P19793 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10822090 0.76 BRD4 (0.43) BRD4XDHBACE1CTSDNOTUM
SCHEMBL5868948 0.71 HCAR3 (0.42) BRD4XDHBACE1CTSDNOTUM
SCHEMBL9198201 0.71 XDH (0.45) TSHRMAPK1BRD4XDHNOTUM
SCHEMBL6996080 0.71 KIF11 (0.44) PTGS1PTGS2KIF11
SCHEMBL10850893 0.70 BRD4 (0.43) TSHRMAPK1BRD4XDHNOTUM
SCHEMBL6997650 0.70 PTGS2 (0.38) BRD4BACE1CTSDNOTUMPGR
SCHEMBL10849821 0.70 XDH (0.47) TSHRMAPK1BRD4XDHNOTUM
SCHEMBL10822086 0.69 BRD4 (0.40) BRD4XDHNOTUMIKBKBPGR
SCHEMBL27564930 0.69 HCAR3 (0.41) BRD4XDHNOTUMIKBKBPGR
SCHEMBL3789224 0.69 TSHR (0.76) TSHRMAPK1BRD4XDHNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3120265-A None JP disclosed
JP-H03120265-A 5H-FURAN-2-ONE DERIVATIVE BAYER AG 1991-05-22 JP disclosed