SCHEMBL9834816

SCHEMBL9834816

CCCOc1ccnc(CSc2nc3ccccc3[nH]2)c1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.58
KMT2A Q03164 4/20 0.58
MEN1 O00255 3/20 0.58
MAPT P10636 3/20 0.58
HTT P42858 3/20 0.58
GALR3 O60755 1/20 0.58
STAT3 P40763 1/20 0.58
NPC1 O15118 7/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2D6 P10635 2/20 0.57
CYP2C9 P11712 2/20 0.57
CYP2C19 P33261 2/20 0.57
CYP3A4 P08684 1/20 0.57
NOS3 P29474 1/20 0.54
NOS1 P29475 1/20 0.54
NOS2 P35228 1/20 0.54
SMN1; SMN2 Q16637 6/20 0.54
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835001 0.91 RAB9A (0.59) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL9833507 0.90 SMN1; SMN2 (0.62) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL6377287 0.87 RAB9A (0.62) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL2992736 0.87 RAB9A (0.74) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL9836498 0.85 RAB9A (0.78) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL6377443 0.85 RAB9A (0.66) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL9834875 0.84 RAB9A (0.66) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL9274369 0.83 NOS3 (0.54) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL8309208 0.82 RAB9A (0.62) RAB9AKMT2AMEN1MAPTHTT
SCHEMBL6377337 0.82 NOS3 (0.58) RAB9AKMT2AMEN1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4738975-A Pyridine derivatives, and use as anti-ulcer agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-04-19 US claimed
EP-0208452-B1 PYRIDINE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1991-09-18 EP disclosed
US-4738975-A Pyridine derivatives, and use as anti-ulcer agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-04-19 US disclosed
EP-0208452-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-01-14 EP disclosed