SCHEMBL9834883

SCHEMBL9834883

CC1(C)C(=O)Nc2cc(NC(=O)C(F)(F)F)c([N+](=O)[O-])cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.40
PDK1 Q15118 2/20 0.38
PDK2 Q15119 2/20 0.38
PDK3 Q15120 2/20 0.38
PDK4 Q16654 2/20 0.38
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
AR P10275 2/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP3A4 P08684 1/20 0.34
ALDH1A1 P00352 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
RECQL P46063 1/20 0.33
GAA P10253 1/20 0.33
THRB P10828 1/20 0.33
HTT P42858 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833300 0.85 NPSR1 (0.45) PGRMEN1KMT2AALDH1A1GAA
SCHEMBL10665255 0.82 ALDH1A1 (0.41) PGRARMEN1KMT2ACYP3A4
SCHEMBL2488888 0.80 NPSR1 (0.45) PGRMEN1KMT2AALDH1A1GAA
SCHEMBL10662304 0.80 HTT (0.52) PGRMEN1KMT2AALDH1A1L3MBTL1
SCHEMBL10376118 0.79 HCAR3 (0.53) PGRMEN1KMT2AALDH1A1GAA
SCHEMBL9833023 0.77 POLB (0.43) MEN1KMT2AALDH1A1RECQLGAA
SCHEMBL10566877 0.76 SMN1; SMN2 (0.58) MEN1KMT2AALDH1A1GAATHRB
SCHEMBL9833900 0.76 AURKB (0.45) PGRMEN1KMT2AALDH1A1GAA
SCHEMBL9559318 0.74 PGR (0.48) PGRPDK2PDK4MEN1KMT2A
SCHEMBL2554351 0.74 RECQL (0.52) PDK1PDK2PDK3PDK4ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed