SCHEMBL9835355

SCHEMBL9835355

CCn1ncc2c(Cl)c(C(=O)c3ccc(OC)cc3)cnc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 5/20 0.55
NR3C1 P04150 6/20 0.53
PGR P06401 1/20 0.49
PDE5A O76074 1/20 0.46
ALDH1A1 P00352 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 1/20 0.45
PDE10A Q9Y233 1/20 0.44
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MAT2A P31153 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 1/20 0.43
ALOX15 P16050 1/20 0.43
PDE1A P54750 1/20 0.43
PDE1B Q01064 1/20 0.43
PDE1C Q14123 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835287 0.88 NR3C1 (0.67) PDE4BNR3C1PGR
SCHEMBL10759905 0.87 PDE4B (0.56) PDE4BNR3C1PDE5AALDH1A1SMN1; SMN2
SCHEMBL9834161 0.87 PDE4B (0.60) PDE4BNR3C1PGRPDE5AMAPT
SCHEMBL9833323 0.87 NR3C1 (0.53) PDE4BNR3C1PGRPDE5AALDH1A1
SCHEMBL9836172 0.86 NR3C1 (0.55) PDE4BNR3C1PGRPDE5A
SCHEMBL9835965 0.86 NR3C1 (0.60) PDE4BNR3C1PGRPDE5A
SCHEMBL5260422 0.85 LMNA (0.50) NR3C1ALDH1A1SMN1; SMN2MAPTNPSR1
SCHEMBL9834731 0.83 NR3C1 (0.55) PDE4BNR3C1PGRALDH1A1MAPT
SCHEMBL4346173 0.82 NR3C1 (0.81) PDE4BNR3C1PGRPDE5A
SCHEMBL9836690 0.81 NR3C1 (0.55) PDE4BNR3C1PGRPDE5APDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230016-B1 6H-Isoxazolo[3,4-d]pyrazolo[3,4-b]pyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-09-11 EP disclosed