SCHEMBL9836285

SCHEMBL9836285

C=CC(=O)NC(C)c1ccccc1S(C)(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 2/20 0.41
TSHR P16473 1/20 0.41
ACACB O00763 2/20 0.40
BCAT2 O15382 1/20 0.37
CYP2C19 P33261 2/20 0.36
CYP3A4 P08684 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP2C9 P11712 1/20 0.36
HTT P42858 1/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
MMP1 P03956 2/20 0.34
MMP2 P08253 2/20 0.34
MMP9 P14780 2/20 0.34
MMP8 P22894 2/20 0.34
MMP12 P39900 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28030413 0.84 TSHR (0.52) TGM2TSHRACACBCYP2C19CYP3A4
SCHEMBL5471473 0.78 TSHR (0.46) TGM2TSHRACACBCYP2C19CYP3A4
SCHEMBL28415923 0.77 TSHR (0.44) TGM2TSHRACACBCYP2C19CYP3A4
Hydrochloric Acid SCHEMBL29110628 0.75 TSHR (0.43) TGM2TSHRACACBCYP2C19CYP3A4
SCHEMBL69176 0.75 LMNA (0.56) CYP2C9
SCHEMBL1330502 0.75 LMNA (0.56) CYP2C9
SCHEMBL4415392 0.73 TDP1 (0.63) TSHRACACBTDP1ALDH1A1MMP9
SCHEMBL5527681 0.73 TDP1 (0.63) TSHRACACBTDP1ALDH1A1MMP9
SCHEMBL28207649 0.73 TDP1 (0.63) TSHRACACBTDP1ALDH1A1MMP9
SCHEMBL28638162 0.71 TGM2 (0.37) TGM2TSHRACACBCYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0272684-B1 DERIVATIVES OF N-(METHYLSULPHONYLPHENYLETHYL)-2-PROPENAMIDES AND THEIR USE AS ANTIBIOTICS ZAMBON S.p.A. (IT) 1991-06-12 EP disclosed
EP-0272684-A2 Derivatives of N-(methylsulphonylphenylethyl)-2-propenamides and their use as antibiotics ZAMBON S.p.A. (IT) 1988-06-29 EP disclosed