SCHEMBL9837623

SCHEMBL9837623

O=c1c2ccc(O)c(Cl)c2oc2cccc(Cl)c12

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 8/20 0.54
EGFR P00533 1/20 0.54
TTR P02766 3/20 0.51
KDM5A P29375 1/20 0.49
PTGS2 P35354 1/20 0.48
ESR1 P03372 4/20 0.47
ESR2 Q92731 4/20 0.47
ATP1A1 P05023 2/20 0.44
ATP1B1 P05026 2/20 0.44
ATP1A3 P13637 2/20 0.44
ATP1B2 P14415 2/20 0.44
ATP1A2 P50993 2/20 0.44
ATP1B3 P54709 2/20 0.44
FXYD2 P54710 2/20 0.44
ATP1A4 Q13733 2/20 0.44
ACE P12821 1/20 0.44
CSNK2A2 P19784 1/20 0.43
CSNK2B P67870 1/20 0.43
CSNK2A1 P68400 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837184 0.85 ESR1 (0.52) MAOAEGFRKDM5APTGS2ESR1
SCHEMBL9836624 0.81 PTGS2 (0.71) MAOAEGFRTTRKDM5APTGS2
SCHEMBL9837036 0.81 ATP1A1 (0.55) MAOAEGFRTTRPTGS2ESR1
SCHEMBL9836052 0.79 SRD5A1 (0.47) MAOAEGFRTTRKDM5APTGS2
SCHEMBL15346134 0.78 ATP1A1 (0.64) MAOAPTGS2ESR1ESR2ATP1A1
SCHEMBL9835732 0.75 TTR (0.48) MAOATTR
SCHEMBL29755034 0.74 KDM4E (0.52) MAOATTRKDM5APTGS2ESR1
SCHEMBL9836803 0.74 TTR (0.54) MAOATTRPTGS2ESR1ESR2
SCHEMBL149545 0.73 MAOA (0.73) MAOAEGFRKDM5APTGS2ATP1A1
SCHEMBL9834846 0.73 AHR (0.54) TTRPTGS2ESR1ESR2ATP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0175376-B1 XANTHONE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME Chugai Seiyaku Kabushiki Kaisha (JP) 1991-04-03 EP disclosed
US-4816479-A HYPOTENSIVE AGENTS, DIURETICS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1989-03-28 US disclosed
US-4661607-A ANTIEDEMIC AGENTS, HYPOTENSIVE AGENTS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1987-04-28 US disclosed
EP-0175376-A2 Xanthone derivatives and process for producing the same Chugai Seiyaku Kabushiki Kaisha (JP) 1986-03-26 EP disclosed