SCHEMBL9838699

SCHEMBL9838699

O=C(O)c1cn(C2CC2)c2nc(N3CC4CCC3CN4CCO)c(F)cc2c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.55
CHRM2 P08172 1/20 0.53
DRD1 P21728 1/20 0.53
LMNA P02545 4/20 0.49
KDM4E B2RXH2 3/20 0.49
HSD17B10 Q99714 3/20 0.49
ABCC4 O15439 1/20 0.49
DHFR P00374 1/20 0.45
TOP2A P11388 5/20 0.44
TOP2B Q02880 5/20 0.44
CYP2C9 P11712 2/20 0.42
ATP6V1B2 P21281 1/20 0.42
TBXA2R P21731 1/20 0.42
EDNRA P25101 1/20 0.42
TARBP2 Q15633 1/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
MAPT P10636 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837575 0.84 DPP4 (0.55) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9867142 0.84 DPP4 (0.56) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9838619 0.83 DPP4 (0.56) DPP4CHRM2DRD1LMNAKDM4E
Hydrochloric Acid SCHEMBL9838610 0.82 DPP4 (0.56) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9686492 0.81 DHFR (0.59) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9837392 0.81 LMNA (0.61) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9668899 0.81 DPP4 (0.60) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9672074 0.81 DPP4 (0.61) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9670599 0.80 DPP4 (0.60) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL9670589 0.79 DPP4 (0.59) DPP4CHRM2DRD1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0159174-B1 SUBSTITUTED NAPHTHYRIDINE-, QUINOLINE- AND BENZOXAZINE- CARBOXYLIC ACIDS AS ANTIBACTERIAL AGENTS AND PROCESSES FOR THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1991-10-23 EP disclosed
US-4571396-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1986-02-18 US disclosed
EP-0159174-A2 Substituted naphthyridine-, quinoline- and benzoxazine- carboxylic acids as antibacterial agents and processes for their production WARNER-LAMBERT COMPANY (US) 1985-10-23 EP disclosed