SCHEMBL9838795

SCHEMBL9838795

Nc1nc2ncc(C=O)cc2c(=O)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NOS1 P29475 6/20 0.43
PNP P00491 2/20 0.41
GART P22102 1/20 0.40
TYMS P04818 2/20 0.39
AKR1B1 P15121 1/20 0.39
DHFR P00374 1/20 0.39
ATIC P31939 1/20 0.39
QTRT1 Q9BXR0 1/20 0.39
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10813052 0.78 CYP1A2 (0.59) CYP1A2KDM4EMEN1ALDH1A1MAPT
SCHEMBL13916085 0.78 CYP1A2 (0.51) CYP1A2KDM4EMEN1ALDH1A1MAPT
SCHEMBL10808383 0.77 CYP1A2 (0.48) CYP1A2KDM4EMEN1ALDH1A1MAPT
SCHEMBL10809113 0.77 GART (0.48) CYP1A2KDM4EMEN1ALDH1A1MAPT
SCHEMBL744451 0.74 CYP1A2 (0.48) CYP1A2KDM4EMEN1ALDH1A1MAPT
SCHEMBL9838375 0.74 KDM4E (0.51) KDM4EMEN1ALDH1A1HPGDKMT2A
SCHEMBL6303945 0.72 DHFR (0.48) DHFR
Hydrochloric Acid SCHEMBL10807714 0.71 DHFR (0.47) DHFR
SCHEMBL13833239 0.70 KDM4E (0.49) CYP1A2KDM4EMEN1ALDH1A1MAPT
SCHEMBL398501 0.70 NOS1 (0.55) KDM4EMEN1ALDH1A1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255228-B1 4(3H)-OXO-5,6,7,8,-TETRAHYDROPYRIDO-(2,3-D)PYRIMIDINE DERIVATIVES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-05-02 EP disclosed
US-4833145-A 4(3H)-oxo-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidine derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-05-23 US disclosed
US-4831037-A 4 (3H)-oxo-5,6,7,8-tetrahydropyrido-(2,3-d)pyrimidine derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-05-16 US disclosed
EP-0255228-A1 4(3H)-Oxo-5,6,7,8,-Tetrahydropyrido-(2,3-d)Pyrimidine derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1988-02-03 EP disclosed