SCHEMBL9840492

SCHEMBL9840492

CON1CCN(C(=O)[C@H](CCC(N)=O)NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
ITGB3 P05106 10/20 0.42
ITGA2B P08514 10/20 0.42
TGM2 P21980 1/20 0.39
HRH2 P25021 3/20 0.38
HRH1 P35367 3/20 0.38
P2RY12 Q9H244 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9840610 0.88 TSHR (0.44) TSHRITGB3ITGA2BTGM2HRH2
SCHEMBL2585311 0.85 P2RY12 (0.50) TSHRITGB3ITGA2BP2RY12
SCHEMBL2585308 0.85 P2RY12 (0.50) TSHRITGB3ITGA2BP2RY12
SCHEMBL9840764 0.80 TGM2 (0.47) TGM2P2RY12KMT2A
SCHEMBL5891360 0.80 CALCRL (0.43) TSHRITGB3ITGA2BHRH2HRH1
SCHEMBL6100308 0.80 PREP (0.52) TSHRITGB3ITGA2B
SCHEMBL18016716 0.79 TSHR (0.44) TSHRITGB3ITGA2BHRH2HRH1
SCHEMBL9840695 0.79 BCHE (0.51) ITGB3ITGA2BHRH2HRH1P2RY12
SCHEMBL6809194 0.78 TSHR (0.41) TSHRITGB3ITGA2BHRH2HRH1
SCHEMBL23326162 0.77 ITGB3 (0.48) TSHRITGB3ITGA2BHRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990614-A N-heterocyclic amides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-02-05 US disclosed
EP-0311517-A2 Amide compound having glutamate receptor inhibiting activity Takeda Chemical Industries, Ltd. (JP) 1989-04-12 EP disclosed