SCHEMBL9844763

SCHEMBL9844763

COC(=O)c1ccc(C=Cc2cn(C)c3nc(N)n(COC(C)C)c(=O)c23)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.36
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 6/20 0.35
TSHR P16473 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
DRD2 P14416 1/20 0.35
PTPN1 P18031 1/20 0.34
TLR8 Q9NR97 1/20 0.34
ADORA2A P29274 2/20 0.33
ADORA2B P29275 2/20 0.33
LMNA P02545 4/20 0.33
MAPT P10636 3/20 0.33
HPGD P15428 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844745 0.90 MAPT (0.35) NPC1RAB9AALDH1A1TSHRSMN1; SMN2
SCHEMBL2072670 0.86 DRD2 (0.40) NPC1RAB9AALDH1A1DRD2PTPN1
SCHEMBL1386593 0.86 DRD2 (0.40) NPC1RAB9AALDH1A1DRD2PTPN1
SCHEMBL9844937 0.72 PTPN1 (0.41) NPC1RAB9AALDH1A1TSHRPTPN1
SCHEMBL9844938 0.72 PTPN1 (0.41) NPC1RAB9AALDH1A1TSHRPTPN1
SCHEMBL8997195 0.66 ATIC (0.35) MAPTKMT2ATP53MEN1TLR7
SCHEMBL71401 0.63 PTPN1 (0.73) NPC1RAB9AALDH1A1TSHRPTPN1
SCHEMBL5379059 0.63 PTPN1 (0.73) NPC1RAB9AALDH1A1TSHRPTPN1
SCHEMBL71402 0.63 PTPN1 (0.73) NPC1RAB9AALDH1A1TSHRPTPN1
SCHEMBL2627847 0.63 PTPN1 (0.73) NPC1RAB9AALDH1A1TSHRPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed