SCHEMBL9844794

SCHEMBL9844794

CN1CC(CCc2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc2)c2c(N)ncnc21

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.51
ATIC P31939 3/20 0.51
GART P22102 7/20 0.49
TYMS P04818 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844818 0.95 DHFR (0.54) DHFRATICGART
SCHEMBL9844736 0.91 GART (0.49) DHFRATICGARTTYMS
SCHEMBL9844836 0.86 DHFR (0.47) DHFRATICGART
SCHEMBL9844885 0.84 ATIC (0.51) DHFRATICGARTTYMS
SCHEMBL9844754 0.84 ATIC (0.51) DHFRATICGARTTYMS
SCHEMBL9844879 0.82 ATIC (0.48) DHFRATICGARTTYMS
SCHEMBL9844814 0.80 DHFR (0.52) DHFRATICGARTTYMS
SCHEMBL9844789 0.77 GART (0.48) DHFRATICGARTTYMS
SCHEMBL8571475 0.74 DHFR (0.57) DHFRGART
SCHEMBL9844757 0.74 DHFR (0.55) DHFRATICGARTTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed