SCHEMBL9845246

SCHEMBL9845246

CC(=O)Nc1ncc2c(ncn2COCC(COC(C)C)OCc2ccccc2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.36
BRD4 O60885 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CYP2C9 P11712 3/20 0.32
CYP2C19 P33261 3/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
GHSR Q92847 1/20 0.32
CYP1A2 P05177 2/20 0.32
ACHE P22303 1/20 0.32
AGER Q15109 1/20 0.32
TSHR P16473 1/20 0.31
FSHR P23945 1/20 0.31
TBXAS1 P24557 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
CCNB2 O95067 1/20 0.31
CCNE2 O96020 1/20 0.31
CDK1 P06493 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9019800 0.93 BCHE (0.38) BCHEBRD4MEN1KMT2ACYP2C9
SCHEMBL9019807 0.85 PDE3A (0.32) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL9575361 0.85 BCHE (0.48) BCHEACHEHPGD
SCHEMBL9019831 0.84 BCHE (0.38) BCHEBRD4MEN1KMT2ACYP2C9
SCHEMBL9019704 0.82 NPR3 (0.40) BCHEBRD4CYP2C9CYP2C19CYP3A4
SCHEMBL9019764 0.81 PDE3A (0.38) MEN1KMT2ACYP2C9CYP2C19CYP3A4
SCHEMBL9575342 0.80 ACHE (0.43) BCHEBRD4MEN1KMT2AACHE
SCHEMBL9845279 0.79 MEN1 (0.39) MEN1KMT2ATSHRMAPK1
SCHEMBL9575434 0.79 CYP1A2 (0.37) BCHEBRD4MEN1KMT2ACYP2C9
SCHEMBL9845278 0.79 SYK (0.31) MEN1KMT2ACYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0452680-A1 Substituted purines, process for their preparation and their use as antiviral agents HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-23 EP disclosed