SCHEMBL9845265

SCHEMBL9845265

CC(=O)Nc1ncc2c(ncn2COCCO)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
HBB P68871 2/20 0.40
PNP P00491 2/20 0.40
USP2 O75604 1/20 0.40
EDNRA P25101 1/20 0.40
HTR2A P28223 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TKT P29401 1/20 0.36
JAK3 P52333 2/20 0.32
JAK1 P23458 1/20 0.32
MAPK1 P28482 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAPK14 Q16539 1/20 0.31
AURKA O14965 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9845279 0.86 MEN1 (0.39) TSHRHBBMEN1KMT2ATKT
SCHEMBL9845272 0.84 CYP3A4 (0.35) TSHRMEN1KMT2ATKT
SCHEMBL9019796 0.82 CYP3A4 (0.41) TSHRBLMMEN1KMT2ATKT
SCHEMBL9845278 0.79 SYK (0.31) TSHRMEN1KMT2A
SCHEMBL9019826 0.77 ALDH1A1 (0.37) TSHRBLMHSD17B10MEN1KMT2A
SCHEMBL9019807 0.77 PDE3A (0.32) BLMMEN1KMT2ATKT
SCHEMBL9019764 0.77 PDE3A (0.38) BLMMEN1KMT2ATKT
SCHEMBL8179334 0.77 TSHR (0.38) TSHRHSD17B10MEN1KMT2AMAPK1
SCHEMBL8172851 0.75 RXFP1 (0.42) TSHRUSP2BLMTKTMAPK1
SCHEMBL9019831 0.74 BCHE (0.38) TSHRBLMMEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0452680-A1 Substituted purines, process for their preparation and their use as antiviral agents HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-23 EP disclosed