SCHEMBL9846107

SCHEMBL9846107

CCc1cc(NCc2c(OC)ccc(C)c2C)c(=O)[nH]c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 4/20 0.41
PDE3A Q14432 4/20 0.41
MAPT P10636 8/20 0.41
KDM4E B2RXH2 5/20 0.39
APAF1 O14727 1/20 0.39
RECQL P46063 1/20 0.39
GAA P10253 5/20 0.39
LMNA P02545 3/20 0.38
ALDH1A1 P00352 2/20 0.38
IDH1 O75874 4/20 0.36
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HPGD P15428 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9170296 0.86 KDM4E (0.44) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9278136 0.81 MAPT (0.51) PDE3BPDE3AMAPTKDM4EGAA
SCHEMBL9846383 0.81 PDE3B (0.43) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL27337641 0.81 POLB (0.49) PDE3BPDE3AMAPTKDM4EGAA
SCHEMBL9846304 0.81 PDE3B (0.41) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9168694 0.80 PDE3B (0.42) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9164330 0.80 MAPT (0.41) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9846165 0.79 PDE3B (0.41) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9283645 0.78 MAPT (0.48) PDE3BPDE3AMAPTKDM4EAPAF1
SCHEMBL9846175 0.78 PDE3B (0.38) PDE3BPDE3AMAPTKDM4EAPAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed