SCHEMBL9846217

SCHEMBL9846217

CCc1cc(COc2cc(CC)c(C)[nH]c2=O)c(OC)nc1C

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 7/20 0.37
PDE3A Q14432 7/20 0.37
POLB P06746 1/20 0.34
HCAR2 Q8TDS4 4/20 0.34
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PDE10A Q9Y233 6/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846113 0.84 P2RX3 (0.34) KDM4EMAPK1
SCHEMBL9846206 0.82 PDE3B (0.40) PDE3BPDE3AHCAR2KDM4EALDH1A1
SCHEMBL9333881 0.77 MAPT (0.35) PDE3BPDE3AHCAR2KDM4EALDH1A1
SCHEMBL9846194 0.74 PDE3B (0.36) PDE3BPDE3AHCAR2KDM4EALDH1A1
SCHEMBL9846195 0.74 PDE3B (0.36) PDE3BPDE3AHCAR2KDM4EALDH1A1
SCHEMBL11894731 0.73 PDE3B (0.35) PDE3BPDE3AHCAR2
SCHEMBL9246249 0.69 MAPT (0.32) PDE3BPDE3AKDM4E
SCHEMBL9272505 0.69 PDE4A (0.40) POLBKDM4EALDH1A1
SCHEMBL9432009 0.69 CD274 (0.38) POLBKDM4EPDE10A
SCHEMBL9281981 0.68 MAPT (0.37) PDE3BPDE3AHCAR2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed