SCHEMBL9846291

SCHEMBL9846291

CCc1cc(C)[nH]c(=O)c1NCc1nc2c(Cl)cccc2o1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.35
PIK3CD O00329 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
IDH1 O75874 1/20 0.33
FABP4 P15090 2/20 0.33
PTGES O14684 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
PIM1 P11309 2/20 0.31
CSNK2A2 P19784 2/20 0.31
CSNK2B P67870 2/20 0.31
PIM3 Q86V86 2/20 0.31
PIM2 Q9P1W9 2/20 0.31
TNKS O95271 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9166348 0.81 IDH1 (0.37) PARP1PIK3CDPIK3CBPIK3CGIDH1
SCHEMBL9846292 0.75 SCN9A (0.35) PARP1PIK3CDPIK3CBPIK3CGIDH1
SCHEMBL9846224 0.73 PARP1 (0.37) PARP1PIK3CDPIK3CBPIK3CGPTGES
SCHEMBL9166681 0.69 PIK3CD (0.41) PARP1PIK3CDPIK3CBPIK3CGIDH1
L-697661 SCHEMBL599639 0.66 FABP4 (0.34) IDH1FABP4ALDH1A1GLAMAPT
L-697661 SCHEMBL29456987 0.66 FABP4 (0.34) IDH1FABP4ALDH1A1GLAMAPT
SCHEMBL9168366 0.65 MTNR1A (0.37) PARP1
SCHEMBL9846171 0.65 MAPT (0.40) PIK3CDPIK3CBALDH1A1GAAMAPT
SCHEMBL9846141 0.64 MAPT (0.38) ALDH1A1GAAMAPTNR4A2F2
SCHEMBL15066674 0.63 SMN1; SMN2 (0.46) ALDH1A1MAPTCYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed