SCHEMBL9846776

SCHEMBL9846776

CC(C)(C)OC(=O)n1c(-c2ccccc2[N+](=O)[O-])c(Br)c2cc(CBr)ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
GSK3B P49841 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42
NR1H2 P55055 7/20 0.36
ALDH1A1 P00352 4/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
NR1H3 Q13133 3/20 0.34
PDE4B Q07343 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
MAPT P10636 1/20 0.34
GAA P10253 2/20 0.33
MET P08581 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846733 0.87 CCNB2 (0.44) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL9846675 0.82 CCNB2 (0.42) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL9846769 0.81 NR1H2 (0.48) NR1H2NR1H3
SCHEMBL9846782 0.76 AGTR1 (0.43)
SCHEMBL3000328 0.76 MCL1 (0.35) NR1H2NR1H3MEN1KMT2A
SCHEMBL9661962 0.76 CCNB2 (0.39) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL3760238 0.76 NR1H2 (0.34) NR1H2ALDH1A1NR1H3MAPT
SCHEMBL9218501 0.75 CCNB2 (0.37) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL10442198 0.75 CHRM2 (0.49) NR1H2NR1H3
SCHEMBL9661956 0.74 CCNB2 (0.37) CCNB2CDK1CCNB1GSK3BCCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429257-A2 Indole derivatives GLAXO GROUP LIMITED (GB) 1991-05-29 EP disclosed