SCHEMBL9846675

SCHEMBL9846675

COC(=O)c1ccccc1-c1c(Br)c2cc(CBr)ccc2n1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 1/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
GSK3B P49841 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42
SLC6A3 Q01959 2/20 0.37
NR1H2 P55055 12/20 0.37
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
NR1H3 Q13133 3/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
BRS3 P32247 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846745 0.87 CCNB2 (0.44) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL9846776 0.82 CCNB2 (0.42) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL9846760 0.80 L3MBTL1 (0.42) SLC6A3NR1H2KMT2AHDAC1HDAC6
SCHEMBL9846753 0.80 PTGDR2 (0.38) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL9846792 0.78 AGTR1 (0.44)
SCHEMBL9846741 0.77 AGTR2 (0.52)
SCHEMBL9846790 0.76 AGTR1 (0.44)
SCHEMBL9218501 0.76 CCNB2 (0.37) CCNB2CDK1CCNB1GSK3BCCNB3
SCHEMBL10442198 0.76 CHRM2 (0.49) NR1H2NR1H3GABRG2GABRB3GABRA5
SCHEMBL9661962 0.75 CCNB2 (0.39) CCNB2CDK1CCNB1GSK3BCCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429257-A2 Indole derivatives GLAXO GROUP LIMITED (GB) 1991-05-29 EP disclosed