SCHEMBL9847680

SCHEMBL9847680

CC1=CC(c2cccc([N+](=O)[O-])c2)C([N+](=O)[O-])=C(C)N1OC=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.40
TSHR P16473 4/20 0.38
ACHE P22303 1/20 0.38
CACNA1F O60840 3/20 0.38
CACNA1D Q01668 3/20 0.38
CACNA1S Q13698 3/20 0.38
CACNA1C Q13936 3/20 0.38
ADORA3 P0DMS8 1/20 0.38
MAPT P10636 4/20 0.37
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
CYP2D6 P10635 2/20 0.36
NFKB1 P19838 2/20 0.36
GMNN O75496 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9847682 0.78 CACNA1F (0.41) LMNATSHRACHECACNA1FCACNA1D
SCHEMBL9847685 0.71 CACNA1F (0.40) LMNATSHRCACNA1FCACNA1DCACNA1S
SCHEMBL5537883 0.68 LMNA (0.41) LMNATSHRACHECACNA1FCACNA1D
SCHEMBL9827844 0.68 CACNA1C (0.43) LMNATSHRCACNA1FCACNA1DCACNA1S
SCHEMBL10469171 0.67 CYP1A2 (0.58) LMNATSHRCACNA1FCACNA1DCACNA1S
SCHEMBL7400532 0.66 CYP1A2 (0.46) LMNATSHRCACNA1FCACNA1DCACNA1S
SCHEMBL7424638 0.66 CACNA1C (0.48) LMNATSHRCACNA1FCACNA1DCACNA1S
SCHEMBL7417203 0.65 LMNA (0.45) LMNATSHRACHECACNA1FCACNA1D
SCHEMBL31069050 0.64 LMNA (0.46) LMNATSHRACHECACNA1FCACNA1D
SCHEMBL3118873 0.64 CYP1A2 (0.44) LMNATSHRCACNA1FCACNA1DCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432751-A2 Isomers of 1-azabicyclo[2.2.2]oct-3-yl 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-5-nitropyridine-3-carboxylate MARION MERRELL DOW INC. (US) 1991-06-19 EP claimed
EP-0432751-A2 Isomers of 1-azabicyclo[2.2.2]oct-3-yl 1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-5-nitropyridine-3-carboxylate MARION MERRELL DOW INC. (US) 1991-06-19 EP disclosed
US-4975437-A Cardiotonic agent MARION LABORATORIES, INC. (US) 1990-12-04 US disclosed