SCHEMBL9848198

SCHEMBL9848198

C=CN=Cc1onc(-c2ccc(OC)cc2)c1C(=O)CC

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.42
PTGS1 P23219 1/20 0.42
PDE3A Q14432 1/20 0.42
BACE1 P56817 8/20 0.41
GPBAR1 Q8TDU6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9848115 0.69 PTGS2 (0.47) PTGS2PTGS1PDE3A
SCHEMBL2775071 0.66 GAA (0.64) PTGS2BACE1GPBAR1
SCHEMBL9848113 0.65 PTGS2 (0.43) PTGS2PTGS1PDE3A
SCHEMBL2777180 0.65 PTGS2 (0.60) PTGS2PTGS1PDE3ABACE1GPBAR1
SCHEMBL5730289 0.64 MEN1 (0.43) PTGS2PTGS1PDE3AGPBAR1
SCHEMBL7558640 0.64 MEN1 (0.68) PTGS2BACE1GPBAR1
SCHEMBL8880593 0.64 SMN1; SMN2 (0.61)
SCHEMBL2723582 0.64 GPBAR1 (0.62) PTGS2BACE1GPBAR1
SCHEMBL11893877 0.64 ALDH1A1 (0.61) PTGS2PTGS1BACE1GPBAR1
SCHEMBL9848202 0.64 SMN1; SMN2 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0414391-A2 Aminoketone derivatives and use thereof MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-02-27 EP disclosed