SCHEMBL9849210

SCHEMBL9849210

O=[PH](OCc1cccc(CBr)c1)OCc1cccc(CBr)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
IDO1 P14902 8/20 0.36
AGXT P21549 5/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
MAOB P27338 1/20 0.34
F2 P00734 4/20 0.34
PTPRC P08575 1/20 0.33
PTPN1 P18031 1/20 0.33
SLC11A2 P49281 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849212 0.85 CYP4F2 (0.36) TRPA1ALDH1A1TSHRIDO1AGXT
SCHEMBL27370549 0.81 IDO1 (0.58) IDO1AGXTMAOB
SCHEMBL9849327 0.79 TRPA1 (0.39) TRPA1ALDH1A1TSHRIDO1
SCHEMBL9849181 0.79 TAAR1 (0.53) MAOBCYP2D6NOS3NOS1NOS2
SCHEMBL27264275 0.77 IDO1 (0.58) IDO1AGXTMAOBCYP3A4
SCHEMBL29149473 0.77 IDO1 (0.58) IDO1AGXTMAOB
SCHEMBL6257617 0.77 CYP19A1 (0.50) ALDH1A1TSHRMAOBCYP3A4
SCHEMBL9849379 0.77 MMP3 (0.46) F2
SCHEMBL2213709 0.76 ALDH1A1 (0.61) TRPA1ALDH1A1TSHRIDO1AGXT
SCHEMBL348159 0.76 ALDH1A1 (0.61) TRPA1ALDH1A1TSHRIDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421436-A2 Substituted carboxytetrahydroisoquinolines and derivatives thereof having pharmaceutical activity WARNER-LAMBERT COMPANY (US) 1991-04-10 EP disclosed