SCHEMBL9849239

SCHEMBL9849239

CC(CI)c1nc(C2CCCCC2)cc(-c2ccc(F)cc2)c1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 3/20 0.48
DHODH Q02127 3/20 0.42
APP P05067 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTGDR Q13258 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
GCGR P47871 1/20 0.36
MAPK14 Q16539 1/20 0.36
BTK Q06187 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8879043 0.88 HMGCR (0.54) HMGCRDHODHAPPKDM4EMAPT
SCHEMBL9849223 0.82 HMGCR (0.53) HMGCRKDM4EMAPTLMNAHPGD
SCHEMBL9849110 0.78 KMT2A (0.48) DHODHKDM4EMAPTHPGDNPSR1
SCHEMBL8878207 0.75 HMGCR (0.55) HMGCRADORA2AADORA1GCGR
SCHEMBL8949911 0.75 HMGCR (0.53) HMGCRAPPKDM4EMAPTLMNA
SCHEMBL8877873 0.72 HMGCR (0.62) HMGCRAPPADORA2AADORA1GCGR
SCHEMBL9849089 0.71 DHODH (0.40) HMGCRDHODH
SCHEMBL8879993 0.69 HMGCR (0.49) HMGCRDHODHKDM4EMAPTLMNA
SCHEMBL8876720 0.69 HMGCR (0.59) HMGCRAPPADORA2AADORA1GCGR
SCHEMBL9849224 0.69 DHODH (0.45) DHODHGCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0444533-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed