SCHEMBL9849692

SCHEMBL9849692

COC(=O)c1ccc(CCc2c(N)nc(N)nc2O)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.38
DHFR P00374 5/20 0.38
PARP1 P09874 1/20 0.37
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 1/20 0.37
PPARG P37231 1/20 0.37
NCOA2 Q15596 1/20 0.37
NCOA1 Q15788 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
HPGD P15428 3/20 0.36
ATM Q13315 2/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
FOLR1 P15328 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90B1 P14625 1/20 0.33
TP53 P04637 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9850002 0.93 HPGD (0.40) MRGPRX4DHFRPARP1NPSR1LMNA
SCHEMBL9849931 0.93 HPGD (0.43) MRGPRX4DHFRPARP1NPSR1LMNA
SCHEMBL9849766 0.92 HPGD (0.44) MRGPRX4DHFRPARP1NPSR1LMNA
SCHEMBL9849782 0.87 FOLR1 (0.41) MRGPRX4DHFRLMNAATMFOLR1
SCHEMBL9849753 0.80 FOLR1 (0.47) DHFRLMNAFOLR1ALDH1A1CYP2D6
SCHEMBL9849759 0.80 FOLR1 (0.44) DHFRLMNAHPGDATMFOLR1
SCHEMBL9850018 0.79 FOLR1 (0.43) DHFRLMNAHPGDFOLR1ALDH1A1
SCHEMBL9849706 0.79 DHFR (0.34) DHFRNPSR1LMNAPPARGNCOA2
SCHEMBL9849678 0.77 DAO (0.38) DHFRNPSR1ATMFOLR1ALDH1A1
SCHEMBL1368290 0.74 NPSR1 (0.50) MRGPRX4PARP1NPSR1LMNAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415510-A2 L-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-03-06 EP disclosed
US-4920125-A L-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1990-04-24 US disclosed