SCHEMBL9851803

SCHEMBL9851803

S=C1Cn2c(cc3ccccc32)-c2ccccc2N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 6/20 0.39
BRD4 O60885 5/20 0.39
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
MAPT P10636 2/20 0.38
RECQL P46063 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
HTR2A P28223 4/20 0.37
HTR2C P28335 4/20 0.37
NPC1 O15118 1/20 0.34
HSP90AA1 P07900 1/20 0.34
THRB P10828 1/20 0.34
HK1 P19367 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
GALK1 P51570 1/20 0.34
BLM P54132 1/20 0.34
HKDC1 Q2TB90 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9851810 0.85 CHRM1 (0.44) ALDH1A1ALOX12SMN1; SMN2
SCHEMBL4135918 0.82 CREBBP (0.46) CREBBPBRD4HTR1ACCNB2CDK1
SCHEMBL10763517 0.73 KDM4E (0.38) CREBBPBRD4KMT2AKDM4EMEN1
SCHEMBL2421457 0.73 KDM4E (0.49) KMT2AKDM4EMEN1MAPTRECQL
SCHEMBL9851805 0.69 CNR1 (0.44) CREBBPBRD4KMT2AMEN1MAPT
SCHEMBL9851806 0.69 HTR2A (0.40) KMT2AKDM4EMEN1MAPTRECQL
SCHEMBL17073536 0.68 AKT1 (0.44) CREBBPBRD4KMT2AKDM4EMEN1
SCHEMBL10761116 0.68 BRD4 (0.44) CREBBPBRD4KDM4EMAPTHPGD
SCHEMBL20777927 0.66 PIM1 (0.39) CREBBPBRD4KMT2AHTR2AHTR2C
SCHEMBL3690376 0.64 CREBBP (0.32) CREBBPBRD4KMT2AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4914201-A CHEMICAL INTERMEDIATES FOR ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-04-03 US claimed
EP-0406719-A1 4h-indolo(1,2-d)(1,2,4)triazolo (4,3-a)(1,4)benzodiazepines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-09 EP disclosed
US-4914201-A CHEMICAL INTERMEDIATES FOR ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-04-03 US disclosed
US-4914201-A CHEMICAL INTERMEDIATES FOR ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-04-03 US disclosed
US-4897392-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-01-30 US disclosed