SCHEMBL9851810

SCHEMBL9851810

S=C1Cn2c(cc3ccccc32)-c2cc(Cl)ccc2N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 11/20 0.44
ALDH1A1 P00352 1/20 0.44
PKM P14618 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALOX12 P18054 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
DRD3 P35462 2/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
TGM2 P21980 1/20 0.34
CES1 P23141 1/20 0.34
CNR1 P21554 1/20 0.34
NTSR1 P30989 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9851803 0.85 CREBBP (0.39) ALDH1A1ALOX12SMN1; SMN2
SCHEMBL9851805 0.85 CNR1 (0.44) DRD3TGM2CES1CNR1NTSR1
SCHEMBL17522841 0.70 PIK3CA (0.41) NPSR1DRD3DRD2DRD4
SCHEMBL4135918 0.69 CREBBP (0.46)
SCHEMBL10416848 0.68 OPRK1 (0.51) DRD3CNR1OPRK1PDE4D
SCHEMBL11686737 0.66 MEN1 (0.50) CHRM1ALDH1A1PKMHTTNPSR1
SCHEMBL10763517 0.66 KDM4E (0.38) PKMSMN1; SMN2
SCHEMBL9851851 0.65 BRD4 (0.52) ALDH1A1SMN1; SMN2DRD3CNR1OPRK1
SCHEMBL9851806 0.64 HTR2A (0.40) CHRM1ALDH1A1PKMHTTNPSR1
SCHEMBL9269071 0.63 TGM2 (0.42) CHRM1ALDH1A1PKMHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4914201-A CHEMICAL INTERMEDIATES FOR ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-04-03 US claimed
EP-0406719-A1 4h-indolo(1,2-d)(1,2,4)triazolo (4,3-a)(1,4)benzodiazepines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-09 EP disclosed
US-4914201-A CHEMICAL INTERMEDIATES FOR ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-04-03 US disclosed
US-4897392-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1990-01-30 US disclosed