SCHEMBL9856663

SCHEMBL9856663

CCCCc1cccc(CC(CCN(C)C)c2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.44
HRH1 P35367 2/20 0.44
OPRM1 P35372 4/20 0.42
DRD3 P35462 4/20 0.42
DRD2 P14416 3/20 0.42
OPRD1 P41143 3/20 0.42
OPRK1 P41145 3/20 0.42
SIGMAR1 Q99720 4/20 0.42
KCNH2 Q12809 2/20 0.40
TAAR1 Q96RJ0 1/20 0.39
CHRM1 P11229 2/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
DRD1 P21728 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
ADRA1A P35348 1/20 0.39
SLC6A3 Q01959 1/20 0.39
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857027 0.86 HTR2A (0.49) HTR2AHRH1OPRM1DRD3OPRK1
SCHEMBL9856741 0.83 HTR2A (0.49) HTR2AHRH1SIGMAR1TAAR1CHRM1
SCHEMBL9856860 0.81 HTR2A (0.49) HTR2AHRH1SIGMAR1TAAR1CHRM1
SCHEMBL9856702 0.81 TAAR1 (0.49) HTR2AHRH1TAAR1CHRM1CHRM2
SCHEMBL9856740 0.80 HTR2A (0.47) HTR2AHRH1OPRM1DRD3OPRK1
SCHEMBL9857014 0.80 TAAR1 (0.54) HTR2AHRH1TAAR1CHRM1SLC6A2
SCHEMBL9857080 0.79 HTR2A (0.50) HTR2AHRH1SIGMAR1TAAR1CHRM1
SCHEMBL9857074 0.78 CYSLTR2 (0.47) HTR2AHRH1CHRM1SLC6A4BCHE
SCHEMBL9856945 0.78 HTR2A (0.49) HTR2AHRH1SIGMAR1KCNH2TAAR1
SCHEMBL9857075 0.77 CALM1 (0.54) HTR2AHRH1TAAR1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996235-A Selectively inhibiting the uptake of serotonin and norepinephrine ELI LILLY AND COMPANY (US) 1991-02-26 US disclosed