SCHEMBL9857762

SCHEMBL9857762

COC=C(c1ccccc1)c1ccco1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 5/20 0.44
PTGS1 P23219 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
PKM P14618 2/20 0.42
KMT2A Q03164 4/20 0.41
TDP1 Q9NUW8 2/20 0.40
PTPN1 P18031 1/20 0.39
MAOB P27338 1/20 0.38
HTT P42858 1/20 0.38
MAPK1 P28482 2/20 0.38
RAB9A P51151 2/20 0.38
MEN1 O00255 2/20 0.38
POLB P06746 1/20 0.38
THRB P10828 1/20 0.38
APEX1 P27695 1/20 0.38
RECQL P46063 1/20 0.38
KCNK3 O14649 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857756 1.00 ALDH1A1 (0.45) ALDH1A1MAPTSMN1; SMN2PTGS1CES2
SCHEMBL28728329 0.79 TSHR (0.44) ALDH1A1MAPTCES2CES1KMT2A
SCHEMBL7551804 0.74 SMN1; SMN2 (0.49) ALDH1A1MAPTSMN1; SMN2PTGS1CES2
SCHEMBL27882775 0.70 SMN1; SMN2 (0.53) ALDH1A1MAPTSMN1; SMN2PTGS1CES2
SCHEMBL9525610 0.70 SIGMAR1 (0.44) ALDH1A1MAPTSMN1; SMN2PTGS1CES2
SCHEMBL9525605 0.70 SIGMAR1 (0.44) ALDH1A1MAPTSMN1; SMN2PTGS1CES2
SCHEMBL2459083 0.70 ALDH1A1 (0.58) ALDH1A1MAPTSMN1; SMN2PTGS1CES2
SCHEMBL10606928 0.69 CYP1B1 (0.40) ALDH1A1SMN1; SMN2CES2CES1KMT2A
SCHEMBL3857938 0.69 SMN1; SMN2 (0.55) ALDH1A1MAPTSMN1; SMN2PTGS1CES2
SCHEMBL1384938 0.69 SMN1; SMN2 (0.55) ALDH1A1MAPTSMN1; SMN2PTGS1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068248-A Analgesics, antipyretics and antiinflammatory agents MERCK & CO., INC. (US) 1991-11-26 US disclosed
EP-0160408-B1 BENZOTHIOPHENES, THEIR PRODUCTION AND USE, AND COMPOSITIONS CONTAINING THEM MERCK & CO. INC. (US) 1989-08-23 EP disclosed
US-4760086-A N-alkenyl-3-hydroxybenzo[b]thiophene-2-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-07-26 US disclosed
EP-0160408-A1 Benzothiophenes, their production and use, and compositions containing them MERCK & CO. INC. (US) 1985-11-06 EP disclosed