SCHEMBL9525610

SCHEMBL9525610

BrCCC=C(c1ccccc1)c1ccco1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.44
SMN1; SMN2 Q16637 4/20 0.41
GPR52 Q9Y2T5 1/20 0.41
ALDH1A1 P00352 5/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 3/20 0.39
PTGS1 P23219 1/20 0.38
PKM P14618 1/20 0.37
PTPN1 P18031 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 2/20 0.36
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
POLB P06746 1/20 0.36
THRB P10828 1/20 0.36
APEX1 P27695 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525605 1.00 SIGMAR1 (0.44) SIGMAR1SMN1; SMN2GPR52ALDH1A1MAPT
SCHEMBL4535241 0.80 SIGMAR1 (0.47) SIGMAR1PTPN1
SCHEMBL9528603 0.71 CYP19A1 (0.50) ALDH1A1KMT2AMEN1
SCHEMBL7551804 0.71 SMN1; SMN2 (0.49) SMN1; SMN2GPR52ALDH1A1MAPTKMT2A
SCHEMBL9528596 0.71 CYP19A1 (0.50) ALDH1A1KMT2AMEN1
SCHEMBL8671036 0.70 TDP1 (0.45) SIGMAR1GPR52ALDH1A1PTPN1CES2
SCHEMBL8671035 0.70 TDP1 (0.45) SIGMAR1GPR52ALDH1A1PTPN1CES2
SCHEMBL9857762 0.70 ALDH1A1 (0.45) SMN1; SMN2ALDH1A1MAPTKMT2APTGS1
SCHEMBL9857756 0.70 ALDH1A1 (0.45) SMN1; SMN2ALDH1A1MAPTKMT2APTGS1
SCHEMBL8511316 0.70 SIGMAR1 (0.53) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231996-B1 NOVEL AMINO ACID DERIVATIVES NOVO NORDISK A/S (DK) 1993-10-06 EP disclosed
US-4931450-A Amino acid derivatives NOVO INDUSTRI A/S (DK) 1990-06-05 US disclosed
EP-0231996-A2 Novel amino acid derivatives NOVO NORDISK A/S (DK) 1987-08-12 EP disclosed