SCHEMBL9858147

SCHEMBL9858147

O=C(O)Oc1cn(Cc2ccccc2F)nn1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.50
KDM1A O60341 6/20 0.45
ATM Q13315 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 3/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM1B Q8NB78 1/20 0.43
MAPT P10636 2/20 0.43
PKM P14618 1/20 0.43
KDM4E B2RXH2 1/20 0.42
CA5A P35218 1/20 0.42
ROCK2 O75116 1/20 0.41
PAK4 O96013 1/20 0.41
PIM1 P11309 1/20 0.41
GSK3B P49841 1/20 0.41
AURKB Q96GD4 1/20 0.41
CYP19A1 P11511 1/20 0.40
KCNMA1 Q12791 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9858306 0.88 HDAC1 (0.49) HDAC1KDM1AATML3MBTL1ALDH1A1
SCHEMBL9858277 0.85 CA5A (0.59) HDAC1KDM1AALDH1A1KDM4ECA5A
SCHEMBL11116350 0.84 TYR (0.50) KDM1AATML3MBTL1ALDH1A1MEN1
SCHEMBL9858012 0.80 CYP2C19 (0.56) ATMALDH1A1MEN1KMT2AMAPT
SCHEMBL9858144 0.79 CA5A (0.55) HDAC1KDM1AATML3MBTL1ALDH1A1
Hydrochloric Acid SCHEMBL10667411 0.78 CA5A (0.53) HDAC1KDM1AATML3MBTL1ALDH1A1
SCHEMBL30645406 0.75 CA5A (0.72) HDAC1KDM1AATML3MBTL1ALDH1A1
SCHEMBL10667399 0.75 CA5A (0.53) HDAC1KDM1AATML3MBTL1ALDH1A1
SCHEMBL9857405 0.75 CA5A (0.72) HDAC1KDM1AATML3MBTL1ALDH1A1
SCHEMBL7137288 0.73 CA5A (0.65) HDAC1KDM1AALDH1A1KDM4ECA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0199262-B1 FLUORINATED BENZYL TRIAZOLE COMPOUNDS CIBA-GEIGY AG (CH) 1991-02-27 EP disclosed
EP-0199262-A2 Fluorinated benzyl triazole compounds CIBA-GEIGY AG (CH) 1986-10-29 EP disclosed