SCHEMBL9861896

SCHEMBL9861896

CCc1ccc(N)c(C(F)(F)C(F)(F)C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.38
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
TRPA1 O75762 1/20 0.33
PDK2 Q15119 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2A6 P11509 1/20 0.32
SKP2 Q13309 1/20 0.32
SIGMAR1 Q99720 2/20 0.32
TAAR1 Q96RJ0 1/20 0.31
PDE2A O00408 1/20 0.30
SLC6A2 P23975 2/20 0.30
SLC6A4 P31645 2/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861936 0.89 FFAR4 (0.43) FFAR4SMN1; SMN2NOS3NOS1NOS2
SCHEMBL10629358 0.82 FFAR4 (0.56) FFAR4SMN1; SMN2NOS3NOS1NOS2
SCHEMBL9861563 0.79 TRPA1 (0.50) TRPA1PDK2CYP1A2CYP2A6ALDH1A1
SCHEMBL3871240 0.74 SMN1; SMN2 (0.38) FFAR4SMN1; SMN2ALDH1A1
SCHEMBL3187513 0.71 TSHR (0.45) SMN1; SMN2ALDH1A1
SCHEMBL30469492 0.71 TSHR (0.45) SMN1; SMN2ALDH1A1
SCHEMBL30469491 0.69 TSHR (0.44) SMN1; SMN2ALDH1A1
SCHEMBL1050419 0.69 TSHR (0.44) SMN1; SMN2ALDH1A1
SCHEMBL9861314 0.69 MAPT (0.39) FFAR4SMN1; SMN2ALDH1A1
SCHEMBL841623 0.68 NOS3 (0.46) SMN1; SMN2NOS3NOS1NOS2TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed