SCHEMBL9864273

SCHEMBL9864273

CCCC(=O)C(N(C)C)C1(c2cccc(C(F)(F)F)c2)CCC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.46
SLC6A3 Q01959 2/20 0.46
SLC6A2 P23975 2/20 0.46
CCR2 P41597 2/20 0.42
OPRM1 P35372 5/20 0.41
OPRL1 P41146 4/20 0.41
KCNN4 O15554 2/20 0.39
OPRK1 P41145 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM1A O60341 2/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9864288 0.91 SLC6A4 (0.47) SLC6A4SLC6A3SLC6A2CCR2OPRM1
SCHEMBL9863936 0.82 OPRM1 (0.43) SLC6A4SLC6A3SLC6A2OPRM1OPRL1
SCHEMBL9863909 0.76 SLC6A4 (0.46) SLC6A4SLC6A3SLC6A2CCR2OPRM1
SCHEMBL9863865 0.76 SLC6A3 (0.38) SLC6A4SLC6A3SLC6A2OPRM1OPRL1
SCHEMBL9864359 0.76 SLC6A4 (0.48) SLC6A4SLC6A3SLC6A2CCR2OPRM1
SCHEMBL9118387 0.76 SLC6A4 (0.52) SLC6A4SLC6A3SLC6A2CCR2OPRM1
Hydrochloric Acid SCHEMBL9864247 0.76 SLC6A4 (0.46) SLC6A4SLC6A3SLC6A2CCR2OPRM1
SCHEMBL9864358 0.75 SLC6A2 (0.44) SLC6A4SLC6A3SLC6A2OPRM1OPRL1
SCHEMBL9864499 0.75 SLC6A4 (0.51) SLC6A4SLC6A3SLC6A2OPRK1CYP3A4
SCHEMBL9864222 0.73 SLC6A4 (0.44) SLC6A4SLC6A3SLC6A2OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-B1 ARYLCYCLOBUTYLALKYL AMINES AND THEIR USE AS ANTIDEPRESSIVE MEDICINES The Boots Company PLC (GB) 1988-06-08 EP disclosed
EP-0191542-A1 Arylcyclobutylalkyl amines and their use as antidepressive medicines The Boots Company PLC (GB) 1986-08-20 EP disclosed