SCHEMBL9864530

SCHEMBL9864530

C=CC(=O)Nc1ccccc1C#N

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.57
KDM4E B2RXH2 5/20 0.57
L3MBTL1 Q9Y468 3/20 0.54
ALDH1A1 P00352 4/20 0.51
TSHR P16473 1/20 0.51
GLA P06280 1/20 0.51
CYP1A2 P05177 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PDK1 Q15118 1/20 0.50
PDK2 Q15119 1/20 0.50
PDK3 Q15120 1/20 0.50
PDK4 Q16654 1/20 0.50
TGM2 P21980 1/20 0.50
KMT2A Q03164 2/20 0.48
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MEN1 O00255 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HPGD P15428 1/20 0.47
CA12 O43570 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31171944 1.00 GAA (0.57) GAAKDM4EL3MBTL1ALDH1A1TSHR
SCHEMBL31228347 0.81 TGM2 (0.65) KDM4EALDH1A1SMN1; SMN2TGM2
SCHEMBL613090 0.81 TGM2 (0.65) KDM4EALDH1A1SMN1; SMN2TGM2
SCHEMBL6858019 0.80 GAA (0.66) GAAKDM4EL3MBTL1ALDH1A1TSHR
SCHEMBL9659766 0.78 MAOB (0.38) GAAKDM4EL3MBTL1ALDH1A1TSHR
SCHEMBL4766358 0.78 GAA (0.69) GAAKDM4EL3MBTL1ALDH1A1TSHR
SCHEMBL30107521 0.78 GAA (0.64) GAAKDM4EL3MBTL1ALDH1A1TSHR
SCHEMBL6222692 0.78 GAA (0.64) GAAKDM4EL3MBTL1ALDH1A1TSHR
SCHEMBL21808550 0.78 TGM2 (0.50) GAAKDM4EALDH1A1TGM2HPGD
SCHEMBL31596298 0.78 MAPK3 (0.38) GAAKDM4EALDH1A1TGM2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106977474-A One kind substitution benzofurane acrylamide derivative of 2 cyano group 3 and its production and use 四川大学 2017-07-25 CN claimed
CN-106977474-B Substituted 2-cyano-3-phenyl furan-acrylamide derivative and preparation method and application thereof 四川大学 2020-04-07 CN disclosed
US-20190293641-A1 ASSAY IMPERIAL COLLEGE INNOVATIONS, LTD. (GB) 2019-09-26 US disclosed
WO-2018033753-A2 ASSAY IMPERIAL INNOVATIONS LIMITED (GB) 2018-02-22 WO disclosed
CN-106977474-A One kind substitution benzofurane acrylamide derivative of 2 cyano group 3 and its production and use 四川大学 2017-07-25 CN disclosed
EP-0409565-A1 Rubber composition useful for tires SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1991-01-23 EP disclosed