SCHEMBL9864627

SCHEMBL9864627

CCCC(=O)C(N(C)C)C1(c2ccccc2F)CCC1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 5/20 0.38
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
ESR1 P03372 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NOTUM Q6P988 1/20 0.32
OPRL1 P41146 1/20 0.31
MAPT P10636 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9863936 0.82 OPRM1 (0.43) HDAC4SLC6A4SLC6A3OPRL1TP53
SCHEMBL9864358 0.78 SLC6A2 (0.44) SLC6A4SLC6A3ALDH1A1KDM4ELMNA
SCHEMBL9863726 0.76 SLC6A3 (0.53) SLC6A4SLC6A3
SCHEMBL9863865 0.75 SLC6A3 (0.38) SLC6A4SLC6A3ALDH1A1LMNACYP3A4
SCHEMBL9864499 0.74 SLC6A4 (0.51) HDAC4SLC6A4SLC6A3ALDH1A1LMNA
SCHEMBL9864273 0.73 SLC6A4 (0.46) SLC6A4SLC6A3ALDH1A1CYP1A2CYP3A4
SCHEMBL9864222 0.72 SLC6A4 (0.44) SLC6A4SLC6A3ALDH1A1LMNAOPRL1
SCHEMBL27283870 0.72 SLC6A3 (0.55) SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL2142 0.68 SLC6A3 (0.36) HDAC4SLC6A4SLC6A3CYP3A4OPRL1
SCHEMBL9864254 0.68 SLC6A4 (0.49) HDAC4SLC6A4SLC6A3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047432-A Antidepressants THE BOOTS COMPANY PLC (GB) 1991-09-10 US disclosed
US-4925879-A ANTIDEPRESSANTS BOOTS COMPANY, PLC (GB) 1990-05-15 US disclosed
EP-0191542-B1 ARYLCYCLOBUTYLALKYL AMINES AND THEIR USE AS ANTIDEPRESSIVE MEDICINES The Boots Company PLC (GB) 1988-06-08 EP disclosed
EP-0191542-A1 Arylcyclobutylalkyl amines and their use as antidepressive medicines The Boots Company PLC (GB) 1986-08-20 EP disclosed