SCHEMBL9865321

SCHEMBL9865321

Cc1sc(S)nc1CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRR1 P24046 1/20 0.38
GAA P10253 2/20 0.37
KDM4E B2RXH2 3/20 0.36
AGBL2 Q5U5Z8 2/20 0.35
ALDH1A1 P00352 3/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
MAPT P10636 2/20 0.32
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
APEX1 P27695 1/20 0.31
SHMT1 P34896 1/20 0.31
SHMT2 P34897 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRB2 P47870 1/20 0.31
HSD17B10 Q99714 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10673071 0.98 GABRR1 (0.37) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL855931 0.80 SLC6A3 (0.41) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL4093001 0.78 GABRR1 (0.39) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL341456 0.77 GABRR1 (0.42) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL1417449 0.77 NOS1 (0.43) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL9865312 0.77 GABRR1 (0.38) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL9864687 0.76 GABRR1 (0.37) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL10360810 0.76 AGBL2 (0.38) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL5517320 0.74 GABRR1 (0.36) GABRR1GAAKDM4EAGBL2ALDH1A1
SCHEMBL4845295 0.74 ALDH1A1 (0.38) GABRR1GAAKDM4EAGBL2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011938-A Antimicrobials ELI LILLY AND COMPANY (US) 1991-04-30 US disclosed
EP-0194571-B1 HETEROCYCLIC DISULFIDES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1990-11-14 EP disclosed
US-4940718-A BACTERICIDES ELI LILLY AND COMPANY (US) 1990-07-10 US disclosed
US-4902707-A Bicyclic pyrazolidinones, compositions and use ELI LILLY AND COMPANY (US) 1990-02-20 US disclosed
US-4826992-A MICROBIOCIDE INTERMEDIATES ELI LILLY AND COMPANY (US) 1989-05-02 US disclosed
EP-0203722-A1 Bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-12-03 EP disclosed
EP-0203723-A1 2,3-(dihydro)bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-12-03 EP disclosed
EP-0202794-A1 7-Substituted-2,3-(Dihydro) bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-11-26 EP disclosed
EP-0202046-A1 7-Substituted bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-11-20 EP disclosed
EP-0194571-A1 Heterocyclic disulfides, process for their preparation and pharmaceutical preparations containing them HOECHST AKTIENGESELLSCHAFT (DE) 1986-09-17 EP disclosed