SCHEMBL9865544

SCHEMBL9865544

COc1cc2c(cc1OC)CCC(N(Cc1ccccc1)C(=O)c1ccccc1)=C2

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.45
ACHE P22303 4/20 0.45
BCHE P06276 3/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 1/20 0.44
HTT P42858 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
HCRTR2 O43614 3/20 0.41
TSHR P16473 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
HCRTR1 O43613 1/20 0.40
PTGES O14684 1/20 0.40
ALOX5 P09917 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2243227 0.94 NPC1 (0.48) TP53ACHEBCHENPC1RAB9A
SCHEMBL29626697 0.90 ACHE (0.45) ACHEBCHENPC1RAB9AHTT
SCHEMBL9701184 0.85 NPC1 (0.51) ACHENPC1RAB9AHTTKMT2A
SCHEMBL12354613 0.80 NPC1 (0.44) TP53NPC1RAB9AKMT2AMEN1
SCHEMBL12354600 0.77 NPC1 (0.42) NPC1RAB9AKMT2AMEN1MAPT
SCHEMBL28858711 0.74 LMNA (0.39) NPC1RAB9AKMT2AMEN1HCRTR2
SCHEMBL29009654 0.72 TP53 (0.49) TP53ACHEBCHENPC1RAB9A
SCHEMBL14174100 0.70 NPC1 (0.63) TP53NPC1RAB9AKMT2AMEN1
SCHEMBL28211195 0.68 KDM4E (0.43) TP53NPC1RAB9AHTTKMT2A
SCHEMBL13503759 0.68 NPC1 (0.57) TP53NPC1RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047536-A Hexahydrobenzo(A)phenanthridine compounds PURDUE RESEARCH FOUNDATION (US) 1991-09-10 US disclosed