SCHEMBL9865665

SCHEMBL9865665

CCCC[S+]([O-])c1sc(C(=O)c2ccccc2)cc1C#N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HPGD P15428 3/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
DYRK1A Q13627 3/20 0.36
DYRK1B Q9Y463 3/20 0.36
CLK1 P49759 2/20 0.36
CES2 O00748 4/20 0.35
CES1 P23141 4/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CLK2 P49760 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CDK9 P50750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865076 0.88 ALDH1A1 (0.42) ALDH1A1HPGDMAPTKMT2AMEN1
SCHEMBL9864134 0.83 USP7 (0.37) ALDH1A1HPGDDYRK1ADYRK1BCLK1
SCHEMBL9865622 0.82 ALDH1A1 (0.42) ALDH1A1HPGDMAPTKMT2AMEN1
SCHEMBL9864903 0.76 ALDH1A1 (0.50) ALDH1A1HPGDMAPTKMT2AMEN1
SCHEMBL9876796 0.73
SCHEMBL10570230 0.71 NPC1 (0.48) ALDH1A1MAPTKMT2AMEN1DYRK1A
SCHEMBL9865184 0.70 USP7 (0.39) ALDH1A1HPGDMAPTKMT2AMEN1
SCHEMBL9865338 0.67 MEN1 (0.41) ALDH1A1HPGDMAPTKMT2AMEN1
SCHEMBL10566637 0.65 CLK2 (0.44) ALDH1A1MAPTDYRK1ADYRK1BCES2
SCHEMBL10570549 0.65 CDK5 (0.58) ALDH1A1MAPTKMT2AMEN1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994485-A Seed and soil fungi, bacteria DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1991-02-19 US disclosed
EP-0234622-B1 NEW THIO COMPOUNDS HAVING FUNGICIDAL ACTIVITY DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-06-27 EP disclosed
EP-0234622-A1 New thio compounds having fungicidal activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1987-09-02 EP disclosed