SCHEMBL9865746

SCHEMBL9865746

CC(C)(C)OC(=O)NC(CC(=O)NC1N=C(c2ccccc2)c2ccccc2NC1=O)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 13/20 0.69
CCKAR P32238 11/20 0.69
SCN9A Q15858 1/20 0.51
NOTCH1 P46531 1/20 0.49
RBPJ Q06330 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL642206 0.86 CCKBR (0.76) CCKBRCCKARSCN9ANOTCH1RBPJ
SCHEMBL644153 0.85 CCKBR (0.74) CCKBRCCKAR
SCHEMBL8774740 0.85 CCKBR (0.74) CCKBRCCKAR
SCHEMBL5656206 0.85 CCKBR (0.74) CCKBRCCKAR
SCHEMBL9526550 0.81 CCKAR (1.00) CCKBRCCKARSCN9ANOTCH1RBPJ
SCHEMBL9526556 0.81 CCKAR (1.00) CCKBRCCKARSCN9ANOTCH1RBPJ
SCHEMBL8746534 0.81 CCKAR (1.00) CCKBRCCKARSCN9ANOTCH1RBPJ
SCHEMBL8746538 0.81 CCKAR (1.00) CCKBRCCKARSCN9ANOTCH1RBPJ
SCHEMBL643214 0.80 CCKBR (0.63) CCKBRCCKAR
SCHEMBL10409010 0.78 CCKBR (0.65) CCKBRCCKARNOTCH1RBPJ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004741-A Cholecystokinin(CCK); Treating Disorders Of The Gastrointestinal Tract, Central Nervous System And Of The Appetite Of Animals MERCK & CO., INC. (US) 1991-04-02 US disclosed
US-4820834-A Benzodiazepine analogs MERCK & CO., INC. (US) 1989-04-11 US disclosed
EP-0284256-A1 Benzodiazepine analogs MERCK & CO. INC. (US) 1988-09-28 EP disclosed