SCHEMBL9865846

SCHEMBL9865846

CC(=O)N1CCC(C(=O)c2cc(F)ccc2F)CC1

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.55
DPP4 P27487 1/20 0.52
DPP7 Q9UHL4 1/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
HTR1F P30939 1/20 0.52
HSD11B1 P28845 3/20 0.51
MAPT P10636 2/20 0.51
LMNA P02545 1/20 0.51
GAA P10253 1/20 0.51
PKM P14618 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1838212 0.89 MEN1 (0.61) ALDH1A1DPP4DPP7MEN1KMT2A
SCHEMBL10637954 0.87 QDPR (0.49) DPP4DPP7MEN1KMT2AHSD11B1
SCHEMBL10396188 0.85 HTR1F (0.67) ALDH1A1MEN1KMT2AHTR1FMAPT
SCHEMBL10966560 0.84 HSD11B1 (0.50) DPP4DPP7MEN1KMT2AHSD11B1
SCHEMBL229876 0.83 HSD11B1 (0.65) ALDH1A1MEN1KMT2AHSD11B1
SCHEMBL11111271 0.82 HSD11B1 (0.59) MEN1KMT2AHSD11B1LMNA
SCHEMBL10395236 0.81 CPS1 (0.55) ALDH1A1MEN1KMT2AHSD11B1
SCHEMBL6212608 0.79 HSD11B1 (0.74) ALDH1A1HSD11B1LMNAGAA
SCHEMBL11619437 0.79 CPS1 (0.56) MEN1KMT2AHSD11B1
SCHEMBL7413579 0.78 HSD11B1 (0.67) ALDH1A1MEN1KMT2AHTR1FHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5057611-A Intermediates for analgesics HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-10-15 US disclosed
US-4833244-A Ethanobenzazepines HOECHST-ROUSEEL PHARMACEUTICALS INC. (US) 1989-05-23 US disclosed
US-4723009-A USING 1-OXA-6-AZA SPIRO(2,5)OCTANE COMPOUNDS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-02-02 US disclosed
US-4654336-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-03-31 US disclosed
EP-0200052-A2 Ethanobenzazepines, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-11-05 EP disclosed