SCHEMBL9866877

SCHEMBL9866877

CC(COc1ccccc1)N=C(N)NCCCc1c[nH]cn1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.35
MAOA P21397 1/20 0.35
PTGS1 P23219 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
MTNR1A P48039 3/20 0.33
MTNR1B P49286 3/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
CYP2D6 P10635 1/20 0.33
ADRB3 P13945 1/20 0.33
RECQL P46063 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867300 0.82 POLB (0.38) HRH3L3MBTL1MTNR1AMTNR1BADRB1
SCHEMBL9867294 0.82 POLB (0.38) HRH3L3MBTL1MTNR1AMTNR1BADRB1
SCHEMBL9866299 0.81 HRH4 (0.37) HRH3HRH4CYP2D6
SCHEMBL9867357 0.80 SCN5A (0.43) HRH3HRH4L3MBTL1
SCHEMBL9865960 0.80 SCN5A (0.42) HRH3HRH4L3MBTL1RECQL
SCHEMBL9866870 0.79 MTNR1A (0.44) HRH3MAOAPTGS1LMNAL3MBTL1
SCHEMBL9867261 0.77 HRH2 (0.35) HRH4LMNAL3MBTL1CYP2D6
SCHEMBL9866068 0.74 ADRB1 (0.39) LMNAADRB2ADRB1CYP2D6ADRB3
SCHEMBL9866059 0.74 ADRB1 (0.41) LMNAADRB2ADRB1CYP2D6ADRB3
SCHEMBL9828417 0.73 KDM1A (0.47) MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021431-A H-1 antagonist, h-2 agonist for treating hypertension, cardiac disease or arterial occlusion HEUMANN PHARMA GMBH & CO. (DE) 1991-06-04 US disclosed
EP-0199845-A1 Imidazolylalkylguanidin derivatives, process for their preparation and pharmaceutical compositions containing them HEUMANN PHARMA GMBH & CO (DE) 1986-11-05 EP disclosed