SCHEMBL9866902

SCHEMBL9866902

CC(=O)N1CCC(O[Si](C)(C)C)(C(=O)c2ccccc2F)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
RAB9A P51151 1/20 0.43
ALDH1A1 P00352 6/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
USP2 O75604 3/20 0.40
PKM P14618 1/20 0.40
CYP2C19 P33261 3/20 0.39
MAPK1 P28482 2/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 3/20 0.39
TSHR P16473 3/20 0.38
HIF1A Q16665 2/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
MAPT P10636 1/20 0.38
KDM4E B2RXH2 2/20 0.38
HTT P42858 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867176 0.79 ALDH1A1 (0.46) MEN1KMT2ARAB9AALDH1A1CYP3A4
SCHEMBL30545399 0.69 TSHR (0.57) MEN1KMT2AALDH1A1CYP2C9PKM
SCHEMBL19461766 0.69 TSHR (0.57) MEN1KMT2AALDH1A1CYP2C9PKM
SCHEMBL6209336 0.68 PARP1 (0.44) MEN1KMT2ATSHRTP53
SCHEMBL29760817 0.68 PARP1 (0.44) MEN1KMT2ATSHRTP53
SCHEMBL11111271 0.66 HSD11B1 (0.59) MEN1KMT2ACYP2C9CYP2C19KDM4E
SCHEMBL21383779 0.66 CES2 (0.46) MEN1KMT2AALDH1A1CYP2C9PKM
SCHEMBL9192885 0.65 GAA (0.50) MEN1KMT2ARAB9AALDH1A1HPGD
SCHEMBL12869290 0.64 KMT2A (0.49) KMT2AALDH1A1PKMMAPK1TSHR
SCHEMBL9866909 0.63 ALDH1A1 (0.44) MEN1KMT2AALDH1A1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5057611-A Intermediates for analgesics HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-10-15 US disclosed
US-4833244-A Ethanobenzazepines HOECHST-ROUSEEL PHARMACEUTICALS INC. (US) 1989-05-23 US disclosed
US-4723009-A USING 1-OXA-6-AZA SPIRO(2,5)OCTANE COMPOUNDS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-02-02 US disclosed
US-4654336-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-03-31 US disclosed
EP-0200052-A2 Ethanobenzazepines, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-11-05 EP disclosed