SCHEMBL9867712

SCHEMBL9867712

O=C(c1ccccc1F)C1CC(O)CCN1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
ALOX15 P16050 1/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
HSD11B1 P28845 1/20 0.39
CNR2 P34972 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MGLL Q99685 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPK14 Q16539 1/20 0.37
KDM4E B2RXH2 2/20 0.36
OPRM1 P35372 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14231067 0.80 ELANE (0.46) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL14230971 0.80 ELANE (0.46) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL9851969 0.70 HTR3E (0.55) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL29591363 0.70 CES2 (0.56) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL718095 0.70 CES2 (0.56) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL747207 0.70 CTSK (0.38) CNR2MEN1KMT2A
Hydrochloric Acid SCHEMBL10395823 0.69 HTR3E (0.54) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL717435 0.67 CES2 (0.52) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL29990216 0.67 CES2 (0.52) ALDH1A1ALOX15CES2CES1HSD11B1
SCHEMBL4006843 0.67 CES2 (0.52) ALDH1A1ALOX15CES2CES1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5057611-A Intermediates for analgesics HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-10-15 US disclosed
US-4833244-A Ethanobenzazepines HOECHST-ROUSEEL PHARMACEUTICALS INC. (US) 1989-05-23 US disclosed
US-4723009-A USING 1-OXA-6-AZA SPIRO(2,5)OCTANE COMPOUNDS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-02-02 US disclosed
US-4654336-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-03-31 US disclosed
EP-0200052-A2 Ethanobenzazepines, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-11-05 EP disclosed