SCHEMBL9868023

SCHEMBL9868023

COC1(c2cc(F)ccc2F)CC12CCN(C(C)=O)CC2

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 6/20 0.41
PSEN2 P49810 6/20 0.41
APH1B Q8WW43 6/20 0.41
NCSTN Q92542 6/20 0.41
APH1A Q96BI3 6/20 0.41
PSENEN Q9NZ42 6/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP2D6 P10635 2/20 0.40
DPP4 P27487 1/20 0.39
DPP7 Q9UHL4 1/20 0.39
CNR1 P21554 1/20 0.38
AKT1 P31749 1/20 0.37
CYP3A4 P08684 1/20 0.36
RORC P51449 1/20 0.36
KIF11 P52732 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 1/20 0.36
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868197 0.77 PSEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4819807 0.68 PSEN1 (0.78) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9866909 0.68 ALDH1A1 (0.44) ALDH1A1CYP2D6DPP4DPP7CYP3A4
SCHEMBL9868636 0.67 ALDH1A1 (0.43) ALDH1A1CYP2D6DPP4DPP7CYP3A4
SCHEMBL14263409 0.65 CES2 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8067224 0.64 OPRM1 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6952918 0.64 NOTUM (0.59) ALDH1A1DPP4DPP7RORC
SCHEMBL7324875 0.64 DPP4 (0.49) ALDH1A1CYP2D6DPP4DPP7RORC
SCHEMBL18711298 0.63 RORC (0.44) ALDH1A1CYP2D6RORCMAPK1CYP2C19
SCHEMBL7701344 0.62 DPP4 (0.46) ALDH1A1CYP2D6DPP4DPP7CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5057611-A Intermediates for analgesics HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-10-15 US disclosed
US-4833244-A Ethanobenzazepines HOECHST-ROUSEEL PHARMACEUTICALS INC. (US) 1989-05-23 US disclosed
US-4723009-A USING 1-OXA-6-AZA SPIRO(2,5)OCTANE COMPOUNDS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-02-02 US disclosed
US-4654336-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-03-31 US disclosed
EP-0200052-A2 Ethanobenzazepines, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-11-05 EP disclosed