SCHEMBL9869234

SCHEMBL9869234

CN1C(=O)C(NC(=O)c2ccc(I)cc2)=NC(c2ccccc2)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 8/20 0.41
CCKAR P32238 6/20 0.41
CYP2C9 P11712 1/20 0.38
ADORA3 P0DMS8 1/20 0.36
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
EGFR P00533 1/20 0.34
SRC P12931 1/20 0.34
DRD2 P14416 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
GABRA4 P48169 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087130 0.73 KCNH2 (0.49) CYP2C9MAPK1GAAALDH1A1HTT
SCHEMBL9726866 0.70 LRRK2 (0.41) MAPK1EGFRGABRPGABRDGABRA1
SCHEMBL8716727 0.68 CCKAR (0.31) CCKBRCCKAR
SCHEMBL6920408 0.65 CHEK1 (0.36) EGFRSRCGAAHDAC4HDAC7
SCHEMBL1868702 0.64 SETDB1 (0.40) CCKBR
Hydrochloric Acid SCHEMBL7208149 0.64 CHEK1 (0.36) EGFRSRCGAAHDAC4HDAC7
SCHEMBL8977555 0.62 CCKBR (0.81) CCKBRCCKARGABRPGABRDGABRA1
SCHEMBL5718666 0.61 PTPN1 (0.71) POLBHTTMEN1KMT2A
SCHEMBL7103601 0.61 MEN1 (0.68) POLBMAPK1MEN1KMT2A
SCHEMBL9704603 0.59 OPRK1 (0.42) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994258-A Radiolabeled cholecystokinin-A antagonists bind to receptors MERCK & CO., INC. (US) 1991-02-19 US disclosed