SCHEMBL9869415

SCHEMBL9869415

COC(=O)c1ccncc1SCc1ccc(OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.53
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
TP53 P04637 2/20 0.45
NOD2 Q9HC29 1/20 0.44
PKM P14618 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
RAB9A P51151 1/20 0.43
FFAR1 O14842 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
RXFP1 Q9HBX9 1/20 0.43
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
KMT2A Q03164 2/20 0.42
DAO P14920 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869063 0.90 LMNA (0.53) LMNAKDM4EALDH1A1GLAGAA
SCHEMBL9869016 0.88 FFAR1 (0.50) LMNAKDM4EGAATP53NOD2
SCHEMBL3780022 0.87 L3MBTL1 (0.59) KDM4EALDH1A1GLAGAATP53
SCHEMBL28326285 0.81 POLB (0.58) LMNAKDM4EALDH1A1TP53PKM
SCHEMBL17080124 0.81 KDM4E (0.52) LMNAKDM4EALDH1A1TP53PKM
SCHEMBL9869231 0.81 FFAR1 (0.50) LMNAKDM4EALDH1A1GAATP53
SCHEMBL17080148 0.79 KDM4E (0.56) LMNAKDM4EALDH1A1TP53PKM
SCHEMBL17080182 0.78 KDM4E (0.46) LMNAKDM4EALDH1A1TP53PKM
SCHEMBL17080139 0.78 CA1 (0.51) LMNAKDM4EALDH1A1GLAGAA
SCHEMBL17080153 0.77 MAPT (0.46) LMNAKDM4EALDH1A1GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006532-A Enzyme inhibitor; antiinflammatory agents MERCK & CO. INC., INC. (US) 1991-04-09 US disclosed
US-4904672-A Derivatives of 3-hydroxyazabenzo[b]thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1990-02-27 US disclosed
US-4767766-A Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-08-30 US disclosed